SCHEMBL20121537

SCHEMBL20121537

CC(C)(C)OC(=O)N[C@@H](Cc1ccc(NO)cc1)C(=O)N1CCn2c(nc(-c3cccc(F)c3)c2Nc2ccc(Cl)c(F)c2)C1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.53
PABPC1 P11940 1/20 0.39
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
MC4R P32245 1/20 0.35
PARP1 P09874 1/20 0.35
P2RX7 Q99572 1/20 0.35
KMT2A Q03164 2/20 0.35
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
ADORA1 P30542 1/20 0.34
PTPRB P23467 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2068538 0.94 KCNH2 (0.54) KCNH2PABPC1CTSSCTSKMC4R
SCHEMBL2069062 0.93 KCNH2 (0.51) KCNH2PABPC1CTSSCTSKMC4R
SCHEMBL2070632 0.92 KCNH2 (0.52) KCNH2PABPC1CTSSCTSKPARP1
SCHEMBL2068274 0.90 KCNH2 (0.48) KCNH2PABPC1CTSSCTSKMC4R
SCHEMBL2068837 0.90 KCNH2 (0.55) KCNH2PABPC1CTSSCTSKMC4R
SCHEMBL18136315 0.87 KCNH2 (0.51) KCNH2PABPC1CTSSCTSKKMT2A
SCHEMBL2070460 0.86 KCNH2 (0.51) KCNH2PABPC1CTSSCTSKP2RX7
SCHEMBL1049662 0.86 KCNH2 (0.62) KCNH2PABPC1CTSSCTSKP2RX7
SCHEMBL2068262 0.86 KCNH2 (0.52) KCNH2PABPC1CTSSCTSKMC4R
SCHEMBL15340404 0.85 KCNH2 (0.58) KCNH2PABPC1CTSSCTSKP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed