SCHEMBL20121551

SCHEMBL20121551

CC(C)CCC(=O)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(F)c(F)c2)C1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.69
CYP3A4 P08684 1/20 0.44
DPP4 P27487 1/20 0.39
DPP8 Q6V1X1 1/20 0.39
CSNK1D P48730 2/20 0.37
CSNK1E P49674 2/20 0.37
TGFBR1 P36897 2/20 0.36
P2RX7 Q99572 1/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12952293 0.93 KCNH2 (0.70) KCNH2CYP3A4DPP4DPP8CSNK1D
SCHEMBL12952177 0.93 KCNH2 (0.77) KCNH2CYP3A4DPP4DPP8CSNK1D
SCHEMBL12952188 0.91 KCNH2 (0.71) KCNH2CYP3A4DPP4DPP8
SCHEMBL12952045 0.90 KCNH2 (0.68) KCNH2CYP3A4DPP4DPP8CSNK1D
SCHEMBL12951890 0.90 KCNH2 (0.77) KCNH2CYP3A4DPP4DPP8CSNK1D
SCHEMBL20121575 0.88 KCNH2 (0.74) KCNH2CYP3A4DPP4DPP8TGFBR1
SCHEMBL15760207 0.88 KCNH2 (0.72) KCNH2CYP3A4DPP4DPP8CSNK1D
SCHEMBL20121599 0.88 KCNH2 (0.68) KCNH2CYP3A4DPP4DPP8CSNK1D
SCHEMBL12952197 0.87 KCNH2 (0.68) KCNH2CYP3A4DPP4DPP8
SCHEMBL20121595 0.87 KCNH2 (0.67) KCNH2CYP3A4DPP4DPP8CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed