SCHEMBL20121555

SCHEMBL20121555

O=C(CC1CC1)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(F)c(F)c2)C1

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.68
CYP3A4 P08684 1/20 0.43
DPP4 P27487 1/20 0.39
DPP8 Q6V1X1 1/20 0.39
P2RX7 Q99572 2/20 0.37
GRIN2B Q13224 1/20 0.36
DGAT1 O75907 1/20 0.36
SOAT1 P35610 1/20 0.36
RORC P51449 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20121607 0.93 KCNH2 (0.70) KCNH2CYP3A4DPP4DPP8RORC
SCHEMBL20121612 0.92 KCNH2 (0.80) KCNH2CYP3A4P2RX7
SCHEMBL12952192 0.91 KCNH2 (0.69) KCNH2CYP3A4DPP4DPP8P2RX7
SCHEMBL20121606 0.90 KCNH2 (0.68) KCNH2CYP3A4P2RX7
SCHEMBL12952185 0.88 KCNH2 (0.78) KCNH2CYP3A4RORC
SCHEMBL2068029 0.88 KCNH2 (0.85) KCNH2CYP3A4DPP4DPP8P2RX7
SCHEMBL20121575 0.88 KCNH2 (0.74) KCNH2CYP3A4DPP4DPP8P2RX7
SCHEMBL12952111 0.88 KCNH2 (0.67) KCNH2CYP3A4DPP4DPP8P2RX7
SCHEMBL12952187 0.87 KCNH2 (0.70) KCNH2CYP3A4DPP4DPP8
SCHEMBL12952188 0.86 KCNH2 (0.71) KCNH2CYP3A4DPP4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed