SCHEMBL20122645

SCHEMBL20122645

C/C=C/c1cnc(C(C)C)cc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CRHBP P24387 1/20 0.35
CYP2C19 P33261 1/20 0.35
CRHR2 Q13324 1/20 0.35
HRH4 Q9H3N8 1/20 0.33
AR P10275 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19191657 0.82 CYP3A4 (0.36) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL20122631 0.80 CYP3A4 (0.31) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL16454730 0.80 SLC22A12 (0.36) CYP3A4CYP2D6TSHRCYP2C19HRH4
SCHEMBL18948445 0.77 CYP3A4 (0.38) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL24665770 0.75 NOTUM (0.37) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL19190749 0.75 CYP3A4 (0.40) CYP3A4CYP2D6CYP2C19AR
SCHEMBL17808240 0.75 CYP2C9 (0.32)
SCHEMBL25797123 0.74 CYP3A4 (0.36) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL19366825 0.74 CYP3A4 (0.36) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL12299819 0.73 AAK1 (0.35) CYP3A4CYP2D6TSHRCRHBPCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963445-B2 Chemical compounds SYNGENTA LIMITED (GB) 2018-05-08 US disclosed