SCHEMBL20124232

SCHEMBL20124232

C=C(CNCc1ccc(C(C)(C)C)cc1)CNC(=N)N

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 9/20 0.45
NR1H4 Q96RI1 7/20 0.45
ANPEP P15144 1/20 0.43
ERAP2 Q6P179 1/20 0.43
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
HDAC3 O15379 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
CA12 O43570 1/20 0.38
CA7 P43166 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11960433 0.83 EPHX2 (0.51) EPHX2NR1H4ANPEPERAP2CA1
SCHEMBL11954 0.80 EPHX2 (0.59) EPHX2NR1H4CA1CA2HDAC3
SCHEMBL11960431 0.77 HDAC3 (0.56) EPHX2NR1H4ANPEPERAP2CA1
SCHEMBL15125586 0.76 EPHX2 (0.55) EPHX2NR1H4CA1CA2HDAC3
SCHEMBL11960454 0.75 EPHX2 (0.45) EPHX2NR1H4ANPEPERAP2CA1
SCHEMBL11960442 0.75 ANPEP (0.52) EPHX2NR1H4ANPEPERAP2CA1
SCHEMBL11774 0.75 ANPEP (0.56) EPHX2NR1H4ANPEPERAP2CA1
SCHEMBL11960455 0.75 BCHE (0.59) EPHX2NR1H4ANPEPERAP2CA1
SCHEMBL11960452 0.74 ANPEP (0.51) EPHX2NR1H4ANPEPERAP2CA1
SCHEMBL11981562 0.72 ANPEP (0.49) EPHX2NR1H4ANPEPERAP2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488532-B1 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME MELINTA THERAPEUTICS INC (US) 2018-05-09 EP disclosed