SCHEMBL20124512

SCHEMBL20124512

Cc1ccnc(CNc2ccc3c(OCCN4CCOCC4)ccc(Cl)c3n2)c1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
TSHR P16473 2/20 0.40
KMO O15229 2/20 0.39
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 2/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
ATM Q13315 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
MAOA P21397 1/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C19 P33261 2/20 0.37
CLK4 Q9HAZ1 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9939693 0.86 NPC1 (0.42) NPC1TSHRKMOALDH1A1KDM4E
SCHEMBL25853966 0.79 NPC1 (0.42) NPC1TSHRKMOMAOAEPHA2
SCHEMBL9939521 0.76 SMN1; SMN2 (0.41) NPC1TSHRKMOALDH1A1KDM4E
SCHEMBL9939180 0.75 TSHR (0.56) NPC1TSHRKMOALDH1A1KDM4E
SCHEMBL22137745 0.73 KDR (0.51) NPC1TSHRALDH1A1KDM4EMAPT
SCHEMBL25854094 0.73 TSHR (0.52) NPC1TSHRKMOALDH1A1KDM4E
SCHEMBL9972390 0.73 KDR (0.56) TSHRMAPTHTR2CHTR2BEPHA2
SCHEMBL9943575 0.73 MAPK14 (0.44) NPC1TSHRKMOALDH1A1KDM4E
SCHEMBL17434796 0.70 ABL1 (0.52) TSHRALDH1A1KDM4E
SCHEMBL17453735 0.70 MAPK14 (0.43) NPC1TSHRALDH1A1KDM4EHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651416-B1 COMPOUNDS USEFUL FOR TREATING AIDS ABIVAX (FR) 2018-05-09 EP disclosed