SCHEMBL20124822

SCHEMBL20124822

Nc1ccc(N2CCCNCC2)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.50
CHRNB2 P17787 7/20 0.48
CHRNA4 P43681 7/20 0.48
HRH3 Q9Y5N1 1/20 0.47
PLD1 Q13393 1/20 0.47
GRIN2D O15399 1/20 0.47
GRIN3B O60391 1/20 0.47
GRIN1 Q05586 1/20 0.47
GRIN2A Q12879 1/20 0.47
GRIN2B Q13224 1/20 0.47
GRIN2C Q14957 1/20 0.47
GRIN3A Q8TCU5 1/20 0.47
CASP1 P29466 1/20 0.44
CASP4 P49662 1/20 0.44
CASP5 P51878 1/20 0.44
UBE2T Q9NPD8 1/20 0.43
PRKCA P17252 1/20 0.43
PRKCQ Q04759 1/20 0.43
PRKCD Q05655 1/20 0.43
BPTF Q12830 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3211478 0.98 HRH4 (0.49) HRH4CHRNB2CHRNA4HRH3PLD1
SCHEMBL31347924 0.93 PLD1 (0.53) HRH4CHRNB2CHRNA4HRH3PLD1
SCHEMBL529383 0.93 PLD1 (0.53) HRH4CHRNB2CHRNA4HRH3PLD1
Hydrochloric Acid SCHEMBL3633878 0.92 PLD1 (0.51) HRH4HRH3PLD1GRIN2DGRIN3B
SCHEMBL29377723 0.84 UBE2T (0.56) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL29739677 0.84 GRIN2D (0.56) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL940331 0.84 GRIN2D (0.56) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL241019 0.84 UBE2T (0.56) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL29739351 0.83 UBE2T (0.54) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL2744803 0.83 UBE2T (0.54) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3008045-B1 ANTIBACTERIAL THIAZOLECARBOXYLIC ACIDS ANTABIO SAS (FR) 2018-05-09 EP disclosed