SCHEMBL20125049

SCHEMBL20125049

Cc1ccc2ncc([N+](=O)[O-])n2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 1.00
CYP2C9 P11712 1/20 1.00
GAA P10253 5/20 0.43
KDM4E B2RXH2 3/20 0.43
GLA P06280 1/20 0.43
ALDH1A1 P00352 7/20 0.40
LMNA P02545 3/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 2/20 0.40
THRB P10828 1/20 0.40
TSHR P16473 1/20 0.40
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
STAT3 P40763 1/20 0.39
CASP3 P42574 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28921245 0.80 CYP1A2 (0.67) CYP1A2CYP2C9GAAALDH1A1LMNA
SCHEMBL18766625 0.80 CYP1A2 (0.67) CYP1A2CYP2C9ALDH1A1LMNAMAPK1
SCHEMBL1356256 0.80 CYP1A2 (0.67) CYP1A2CYP2C9KDM4EALDH1A1LMNA
SCHEMBL5253694 0.80 CYP1A2 (0.67) CYP1A2CYP2C9GAAKDM4EALDH1A1
SCHEMBL15828608 0.80 CYP1A2 (0.66) CYP1A2CYP2C9GAAKDM4EALDH1A1
SCHEMBL18785961 0.73 CYP1A2 (0.56) CYP1A2CYP2C9
SCHEMBL29018907 0.72 CYP1A2 (0.57) CYP1A2CYP2C9ALDH1A1LMNAMAPT
SCHEMBL10238918 0.72 CYP1A2 (0.56) CYP1A2CYP2C9GAAKDM4EGLA
SCHEMBL12789891 0.71 CYP1A2 (0.55) CYP1A2CYP2C9GAAKDM4EGLA
SCHEMBL30217955 0.70 CYP1A2 (0.53) CYP1A2CYP2C9KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3318557-A2 QUINOLONE COMPOUND Otsuka Pharmaceutical Co., Ltd. (JP) 2018-05-09 EP disclosed