Ciglitazone

Ciglitazone

SCHEMBL20125576

CC1(COc2ccc(C[C@H]3SC(=O)NC3=O)cc2)CCCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 1.00
CYP3A4 P08684 2/20 1.00
MAPT P10636 2/20 1.00
MEN1 O00255 1/20 1.00
ALDH1A1 P00352 1/20 1.00
TP53 P04637 1/20 1.00
CYP1A2 P05177 1/20 1.00
ALOX15 P16050 1/20 1.00
TSHR P16473 1/20 1.00
KMT2A Q03164 1/20 1.00
HSD17B10 Q99714 1/20 1.00
TDP1 Q9NUW8 1/20 1.00
HRH3 Q9Y5N1 1/20 0.60
FFAR1 O14842 5/20 0.57
PPARA Q07869 2/20 0.57
PPARG P37231 9/20 0.55
PARP1 P09874 1/20 0.53
RXRA P19793 1/20 0.52
MPC2 O95563 2/20 0.51
CYP2C8 P10632 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ciglitazone SCHEMBL20125581 1.00 HPGD (1.00) HPGDCYP3A4MAPTMEN1ALDH1A1
Ciglitazone SCHEMBL38185 1.00 HPGD (1.00) HPGDCYP3A4MAPTMEN1ALDH1A1
Ciglitazone SCHEMBL21582134 0.99 HPGD (0.98) HPGDCYP3A4MAPTMEN1ALDH1A1
Ciglitazone SCHEMBL3189397 0.99 HPGD (0.98) HPGDCYP3A4MAPTMEN1ALDH1A1
Ciglitazone SCHEMBL8498957 0.94 HPGD (0.89) HPGDCYP3A4MAPTMEN1ALDH1A1
Ciglitazone SCHEMBL6203612 0.92 HPGD (0.84) HPGDCYP3A4MAPTMEN1ALDH1A1
SCHEMBL11091437 0.89 CYP3A4 (0.81) HPGDCYP3A4MAPTMEN1ALDH1A1
SCHEMBL11088249 0.88 CYP3A4 (0.79) HPGDCYP3A4MAPTMEN1ALDH1A1
SCHEMBL12521714 0.88 HPGD (0.79) HPGDCYP3A4MAPTMEN1ALDH1A1
SCHEMBL11083961 0.88 CYP3A4 (0.78) HPGDCYP3A4MAPTMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200253937-A1 5-DEUTERO-THIAZOLIDINE-2,4-DIONE COMPOUNDS AND METHODS OF TREATING MEDICAL DISORDERS USING SAME POXEL SA (FR) 2020-08-13 US disclosed
US-20180125827-A1 5-DEUTERO-THIAZOLIDINE-2,4-DIONE COMPOUNDS AND METHODS OF TREATING MEDICAL DISORDERS USING SAME DEUTERX, LLC 2018-05-10 US disclosed
US-20180125827-A1 5-DEUTERO-THIAZOLIDINE-2,4-DIONE COMPOUNDS AND METHODS OF TREATING MEDICAL DISORDERS USING SAME DEUTERX, LLC 2018-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180125827-A1 5-DEUTERO-THIAZOLIDINE-2,4-DIONE COMPOUNDS AND METHODS OF TREATING MEDICAL DISORDERS USING SAME DPP4, SLC5A2, GLP1R HPGD 567/4885CYP3A4 129/4885MAPT 1719/4885
US-20200253937-A1 5-DEUTERO-THIAZOLIDINE-2,4-DIONE COMPOUNDS AND METHODS OF TREATING MEDICAL DISORDERS USING SAME SLC5A2, GLI2, SLC5A1 HPGD 482/4885CYP3A4 95/4885MAPT 674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.