SCHEMBL20129162

SCHEMBL20129162

c1ccc(COCCOCCOCCOC2CCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
LTA4H P09960 1/20 0.46
FOXM1 Q08050 1/20 0.46
NAAA Q02083 1/20 0.45
LIPG Q9Y5X9 1/20 0.41
OPRM1 P35372 2/20 0.41
OPRL1 P41146 2/20 0.41
DPP4 P27487 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
POLB P06746 1/20 0.40
TMEM97 Q5BJF2 1/20 0.39
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
PRMT8 Q9NR22 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
EPHX2 P34913 1/20 0.39
CYP2C19 P33261 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20129240 1.00 TSHR (0.47) TSHRLTA4HFOXM1NAAALIPG
SCHEMBL21456425 0.98 TSHR (0.48) TSHRLTA4HFOXM1NAAALIPG
SCHEMBL23868167 0.91 TSHR (0.52) TSHRLTA4HNAAALIPGOPRM1
SCHEMBL22787012 0.87 FOXM1 (0.45) TSHRLTA4HFOXM1NAAAOPRM1
SCHEMBL18085580 0.87 TSHR (0.41) TSHRLTA4HFOXM1NAAALIPG
SCHEMBL12561351 0.86 TSHR (0.47) TSHRLTA4HFOXM1OPRM1OPRL1
SCHEMBL22906857 0.85 SLC6A2 (0.49) TSHRNAAA
SCHEMBL578557 0.85 TSHR (0.42) TSHRLTA4HFOXM1NAAALIPG
SCHEMBL23267243 0.85 SLC6A2 (0.49) TSHRNAAA
SCHEMBL23462124 0.83 TSHR (0.44) TSHRLTA4HNAAALIPGOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11912699-B2 Tau-protein targeting compounds and associated ARVINAS OPERATIONS, INC. (US) 2024-02-27 US disclosed
US-20180125821-A1 TAU-PROTEIN TARGETING PROTACS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. 2018-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11912699-B2 Tau-protein targeting compounds and associated MAPT, VHL, CRBN TSHR 4013/4885LTA4H 4411/4885FOXM1 2387/4885
US-20180125821-A1 TAU-PROTEIN TARGETING PROTACS AND ASSOCIATED METHODS OF USE CRBN, VHL, UBQLN2 TSHR 3954/4885LTA4H 4566/4885FOXM1 2329/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.