SCHEMBL20134719

SCHEMBL20134719

CC(C)(C)OC(=O)N1[C@@H](CCCCF)C(=O)O[C@@H](c2ccccc2)[C@@H]1c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.43
RORC P51449 2/20 0.34
KLK7 P49862 6/20 0.33
TACR1 P25103 5/20 0.33
KLK5 Q9Y337 5/20 0.32
PRSS1 P07477 2/20 0.32
PRSS2 P07478 2/20 0.32
PRSS3 P35030 2/20 0.32
NR1H2 P55055 3/20 0.32
RXRA P19793 2/20 0.32
NR1H3 Q13133 2/20 0.32
GPR119 Q8TDV5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18109300 1.00 ABCB1 (0.43) ABCB1RORCKLK7TACR1KLK5
SCHEMBL18109299 1.00 ABCB1 (0.43) ABCB1RORCKLK7TACR1KLK5
SCHEMBL18109332 0.91 ABCB1 (0.43) ABCB1KLK7KLK5PRSS1PRSS2
SCHEMBL18109330 0.91 ABCB1 (0.43) ABCB1KLK7KLK5PRSS1PRSS2
SCHEMBL3717651 0.89 ABCB1 (0.42) ABCB1RORCKLK7KLK5PRSS1
SCHEMBL18109442 0.89 ABCB1 (0.42) ABCB1RORCKLK7TACR1KLK5
SCHEMBL18109438 0.89 ABCB1 (0.42) ABCB1RORCKLK7TACR1KLK5
SCHEMBL19461020 0.89 ABCB1 (0.42) ABCB1RORCKLK7TACR1KLK5
SCHEMBL895150 0.84 ABCB1 (0.40) ABCB1RORCKLK7NR1H2RXRA
SCHEMBL895149 0.84 ABCB1 (0.40) ABCB1RORCKLK7NR1H2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321265-A1 4,6-DIAMINO-PYRIDO[3,2-D]PYRIMIDINE COMPOUNDS AND THEIR UTILISATION AS MODULATORS OF TOLL-LIKE RECEPTORS Gilead Sciences, Inc. (US) 2018-05-16 EP disclosed