SCHEMBL20138694

SCHEMBL20138694

Fc1cc(Cl)cc(Oc2nc(Br)nn2CC2CC(F)C2F)c1

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 7/20 0.32
VEGFA P15692 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20138693 0.80 VEGFA (0.33) EPAS1VEGFA
SCHEMBL20138689 0.78 EPAS1 (0.38) EPAS1VEGFA
SCHEMBL20138687 0.77 EPAS1 (0.39) EPAS1VEGFA
SCHEMBL20142985 0.77 EPAS1 (0.41) EPAS1VEGFA
SCHEMBL20138849 0.77 EPAS1 (0.38) EPAS1VEGFA
SCHEMBL20143018 0.76 EPAS1 (0.37) EPAS1VEGFA
SCHEMBL20138802 0.76 EPAS1 (0.41) EPAS1VEGFA
SCHEMBL20138671 0.75 EPAS1 (0.36) EPAS1VEGFA
SCHEMBL20138674 0.75 EPAS1 (0.37) EPAS1VEGFA
SCHEMBL20154257 0.74 EPAS1 (0.37) EPAS1VEGFA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538516-A1 PHENOXYTRIAZOLES F. Hoffmann-La Roche AG (CH) 2019-09-18 EP disclosed
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed