SCHEMBL20141020

SCHEMBL20141020

Cc1c(CN2CCN(c3ccccc3C#N)CC2)cc(C(=O)N2CCCN(c3cccc(C#N)c3)CC2)n1C

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTOR P42345 6/20 0.68
RPTOR Q8N122 6/20 0.68
MLST8 Q9BVC4 6/20 0.68
DRD2 P14416 3/20 0.44
HTR7 P34969 1/20 0.43
DRD3 P35462 2/20 0.43
CHRM4 P08173 2/20 0.41
DRD4 P21917 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
HTR2A P28223 1/20 0.41
THPO P40225 1/20 0.41
HIF1A Q16665 1/20 0.41
HTR1A P08908 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139510 0.93 MTOR (0.68) MTORRPTORMLST8DRD2DRD3
SCHEMBL20159146 0.91 MTOR (0.68) MTORRPTORMLST8DRD2DRD3
SCHEMBL20158919 0.89 MTOR (0.72) MTORRPTORMLST8DRD2HTR7
SCHEMBL20158992 0.89 MTOR (0.84) MTORRPTORMLST8DRD2HTR7
SCHEMBL20158995 0.88 MTOR (0.74) MTORRPTORMLST8DRD2HTR7
SCHEMBL20159082 0.88 MTOR (0.75) MTORRPTORMLST8DRD2HTR7
SCHEMBL20141378 0.88 MTOR (0.69) MTORRPTORMLST8DRD2HTR7
SCHEMBL20159161 0.84 MTOR (0.64) MTORRPTORMLST8DRD2HTR7
SCHEMBL20158988 0.84 MTOR (0.73) MTORRPTORMLST8DRD2HTR7
SCHEMBL20159090 0.83 MTOR (0.71) MTORRPTORMLST8DRD2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed