SCHEMBL20142845

SCHEMBL20142845

Cc1ccc(Nc2nc(N)c(C(=O)c3ccc(F)cc3)s2)cc1

nearest known ligand 0.79

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.79
MEN1 O00255 4/20 0.79
KMT2A Q03164 4/20 0.79
CCNA2 P20248 7/20 0.78
CDK2 P24941 7/20 0.78
CDK5 Q00535 8/20 0.76
CDK5R1 Q15078 8/20 0.76
MAPT P10636 4/20 0.76
TP53 P04637 2/20 0.76
GSK3A P49840 2/20 0.73
GSK3B P49841 2/20 0.73
LMNA P02545 2/20 0.65
RAB9A P51151 2/20 0.63
MAPK14 Q16539 1/20 0.63
TDP1 Q9NUW8 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25609657 1.00 NPC1 (0.79) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL13633841 0.94 CCNA2 (0.88) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL25611327 0.88 NPC1 (0.76) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL25609654 0.88 MEN1 (1.00) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL20142856 0.88 MEN1 (1.00) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL25610719 0.88 NPC1 (0.76) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL20142192 0.88 CCNA2 (0.78) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL20142403 0.88 CCNA2 (0.78) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL25609762 0.88 CCNA2 (0.78) NPC1MEN1KMT2ACCNA2CDK2
SCHEMBL20142846 0.88 CCNA2 (0.78) NPC1MEN1KMT2ACCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO claimed
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO disclosed