SCHEMBL20143121

SCHEMBL20143121

CC(F)(F)CN1CCCc2cc(O)ccc2C1c1ccc(OCCN2CC(CF)C2)cc1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 20/20 0.58
ESR2 Q92731 2/20 0.54
HDAC6 Q9UBN7 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20143175 1.00 ESR1 (0.58) ESR1ESR2HDAC6
SCHEMBL19439349 0.93 ESR1 (0.60) ESR1ESR2
SCHEMBL19454289 0.93 ESR1 (0.60) ESR1ESR2
SCHEMBL19439321 0.93 ESR1 (0.60) ESR1ESR2
SCHEMBL19454227 0.90 ESR1 (0.65) ESR1ESR2HDAC6
SCHEMBL19454226 0.90 ESR1 (0.65) ESR1ESR2HDAC6
SCHEMBL19454230 0.90 ESR1 (0.65) ESR1ESR2HDAC6
SCHEMBL19439359 0.88 ESR1 (0.61) ESR1ESR2HDAC6
SCHEMBL19439356 0.88 ESR1 (0.61) ESR1ESR2HDAC6
SCHEMBL19439319 0.88 ESR1 (0.61) ESR1ESR2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9969732-B2 Tetrahydroisoquinoline estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2018-05-15 US disclosed