SCHEMBL20143797

SCHEMBL20143797

O=C(O)CN(CCN1CC(=O)OC(=O)C1)CCN1CC(=O)OC(=S)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
CHRM2 P08172 1/20 0.35
ADRA2A P08913 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
DRD1 P21728 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
CYP2C19 P33261 1/20 0.35
ADRA1A P35348 1/20 0.35
DRD3 P35462 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
EYA2 O00167 1/20 0.32
APP P05067 1/20 0.32
ACE P12821 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL124918 0.91 TDP1 (0.42) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL9152846 0.90 TDP1 (0.45) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL110199 0.88 TDP1 (0.48) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL2809739 0.88 TDP1 (0.43) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL12438502 0.84 TDP1 (0.36) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL14488349 0.83 TDP1 (0.39) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL8209723 0.82 TDP1 (0.38) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL15749902 0.82 GLA (0.44) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL15165746 0.81 TDP1 (0.33) TDP1KDM4ELMNACHRM2ADRA2A
SCHEMBL19652368 0.81 TDP1 (0.37) TDP1KDM4ELMNACHRM2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9969681-B2 DTPA prodrugs, compositions thereof, and methods of using the same THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2018-05-15 US disclosed