SCHEMBL20144243

SCHEMBL20144243

CC(C)(C)OC(=O)N1CCC(n2nc(-c3ccc(Oc4ccccc4)cn3)c3c(N)ncnc32)CC1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.64
EGFR P00533 2/20 0.60
LCK P06239 2/20 0.59
ITK Q08881 1/20 0.59
NUDT14 O95848 1/20 0.58
NUDT5 Q9UKK9 1/20 0.58
LYN P07948 1/20 0.54
KIT P10721 1/20 0.53
FLT3 P36888 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21338891 0.91 BTK (0.76) BTKEGFRLCKITKNUDT14
SCHEMBL17951556 0.90 BTK (0.73) BTKEGFRLCKITKNUDT14
SCHEMBL20144246 0.89 BTK (0.60) BTKEGFRLCKITK
SCHEMBL16075002 0.88 BTK (0.76) BTK
SCHEMBL16074999 0.87 BTK (0.77) BTK
SCHEMBL16075001 0.87 BTK (0.77) BTK
SCHEMBL16123023 0.87 BTK (0.77) BTK
SCHEMBL22720698 0.87 BTK (0.69) BTKEGFRLCKITKNUDT14
SCHEMBL22720690 0.87 BTK (0.69) BTKEGFRLCKITKNUDT14
SCHEMBL5801559 0.87 BTK (0.69) BTKEGFRLCKITKNUDT14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970300-B1 HETEROAROMATIC COMPOUNDS AS BTK INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-05-16 EP disclosed