SCHEMBL20144255

SCHEMBL20144255

C=CC(=O)N1CCC(n2nc(-c3ccc(Oc4ccccc4)nc3)c3c(N)ncnc32)CC1

nearest known ligand 0.91

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.91
EGFR P00533 4/20 0.83
BLK P51451 2/20 0.71
TEC P42680 3/20 0.69
BMX P51813 3/20 0.69
TXK P42681 2/20 0.69
LYN P07948 2/20 0.69
FGFR2 P21802 2/20 0.69
ITK Q08881 2/20 0.69
RIPK2 O43353 1/20 0.69
NR1I2 O75469 1/20 0.69
SLC22A3 O75751 1/20 0.69
LATS1 O95835 1/20 0.69
NUDT14 O95848 1/20 0.69
ABL1 P00519 1/20 0.69
ERBB2 P04626 1/20 0.69
LCK P06239 1/20 0.69
FYN P06241 1/20 0.69
PGR P06401 1/20 0.69
CSF1R P07333 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21330628 0.95 BTK (1.00) BTKEGFRBLKTECBMX
SCHEMBL20177256 0.95 BTK (1.00) BTKEGFRBLKTECBMX
SCHEMBL202187 0.91 BTK (1.00) BTKEGFRBLKTECBMX
SCHEMBL30331082 0.91 BTK (0.78) BTKEGFRBLKLYNITK
SCHEMBL21338838 0.91 BTK (0.91) BTKEGFRBLKTECBMX
SCHEMBL21330630 0.91 BTK (0.91) BTKEGFRBLKTECBMX
SCHEMBL20177281 0.91 BTK (0.91) BTKEGFRBLKTECBMX
SCHEMBL20144254 0.91 BTK (0.80) BTKEGFRBLKITKLCK
SCHEMBL16074979 0.88 BTK (1.00) BTKEGFRBLK
SCHEMBL200392 0.86 BTK (1.00) BTKEGFRBLKTECBMX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970300-B1 HETEROAROMATIC COMPOUNDS AS BTK INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-05-16 EP disclosed