SCHEMBL20144712

SCHEMBL20144712

Nc1ccc2c(c1)N(CCNCN1CCCCC1)CCC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.42
BRD4 O60885 1/20 0.39
ATAD2 Q6PL18 1/20 0.39
CHRM2 P08172 2/20 0.38
CHRM4 P08173 2/20 0.38
REN P00797 4/20 0.38
CYP3A4 P08684 3/20 0.38
TRPV1 Q8NER1 1/20 0.36
ALDH1A1 P00352 3/20 0.35
POLB P06746 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NOS3 P29474 3/20 0.34
NOS1 P29475 3/20 0.34
NOS2 P35228 2/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15038011 0.91 HRH3 (0.46) HRH3BRD4ATAD2CHRM2CHRM4
SCHEMBL15038009 0.90 HRH3 (0.44) HRH3BRD4ATAD2CHRM2CHRM4
SCHEMBL15037987 0.88 HRH3 (0.48) HRH3BRD4ATAD2CHRM2CHRM4
SCHEMBL15037984 0.86 HRH3 (0.46) HRH3BRD4ATAD2CHRM2CHRM4
SCHEMBL15037989 0.84 HRH3 (0.50) HRH3BRD4ATAD2CHRM2CHRM4
SCHEMBL15037988 0.83 HRH3 (0.48) HRH3BRD4ATAD2CHRM2CHRM4
SCHEMBL15038010 0.82 KDM1A (0.41) HRH3BRD4ATAD2RENCYP3A4
SCHEMBL20144797 0.81 BRD4 (0.42) HRH3BRD4ATAD2RENCYP3A4
SCHEMBL15038014 0.81 KDM1A (0.42) HRH3BRD4ATAD2RENCYP3A4
SCHEMBL15037985 0.80 HRH3 (0.42) HRH3BRD4ATAD2RENCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2791116-B1 COUPLER WITH 7-AMINO-1,2,3,4-TETRAHYDROQUINOLINE STRUCTURE, DYEING COMPOSITION COMPRISING SAME, PROCESSES AND USES OREAL (FR) 2018-05-16 EP disclosed