SCHEMBL20145111

SCHEMBL20145111

COc1ccc(C(=O)N2CCCC(Nc3ncc(C(F)(F)F)cn3)C2)c(Cl)n1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK12 Q9NYV4 7/20 0.46
EGFR P00533 2/20 0.45
BTK Q06187 1/20 0.45
ITK Q08881 1/20 0.45
CCNK O75909 5/20 0.44
KMT2A Q03164 1/20 0.44
HCRTR1 O43613 3/20 0.43
GAA P10253 1/20 0.43
HCRTR2 O43614 2/20 0.42
MAPK3 P27361 1/20 0.42
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CDK7 P50613 1/20 0.41
CCNH P51946 1/20 0.41
MNAT1 P51948 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20144832 0.90 HCRTR2 (0.45) KMT2AHCRTR1GAAHCRTR2
SCHEMBL20145258 0.90 HCRTR2 (0.45) KMT2AHCRTR1GAAHCRTR2
SCHEMBL16147941 0.82 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL20144834 0.78 HCRTR1 (0.71) HCRTR1GAAHCRTR2
SCHEMBL20144867 0.77 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL20144731 0.76 HCRTR1 (0.71) HCRTR1HCRTR2
SCHEMBL20144982 0.75 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL25226590 0.74 MAPK3 (0.50) CDK12BTKCCNKKMT2AHCRTR1
SCHEMBL16155578 0.74 HCRTR2 (0.67) HCRTR1HCRTR2
SCHEMBL20145032 0.74 HCRTR1 (0.71) CDK12CCNKHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed