SCHEMBL20145185

SCHEMBL20145185

FC(F)(F)c1ccc(N[C@@H]2CCCNC2)nc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IL1B P01584 2/20 0.53
NLRP3 Q96P20 1/20 0.53
PIM1 P11309 1/20 0.50
IDH2 P48735 1/20 0.50
CHEK1 O14757 1/20 0.48
PDPK1 O15530 1/20 0.47
RPS6KB1 P23443 1/20 0.47
CCR6 P51684 3/20 0.46
IRAK4 Q9NWZ3 2/20 0.46
HCRTR1 O43613 1/20 0.46
MAPK1 P28482 1/20 0.45
CCNT1 O60563 1/20 0.44
CCNK O75909 1/20 0.44
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
CDK9 P50750 1/20 0.44
CDK12 Q9NYV4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1033310 0.92 MAPK1 (0.53) IL1BIDH2CCR6HCRTR1MAPK1
SCHEMBL1033312 0.92 MAPK1 (0.53) IL1BIDH2CCR6HCRTR1MAPK1
SCHEMBL6573805 0.92 MAPK1 (0.53) IL1BIDH2CCR6HCRTR1MAPK1
SCHEMBL17741141 0.86 CCR6 (0.48) CCR6HCRTR1MAPK1
Hydrochloric Acid SCHEMBL17729593 0.84 CCR6 (0.47) CCR6HCRTR1MAPK1
SCHEMBL18607634 0.84 CCR6 (0.55) PIM1CCR6HCRTR1CCNKCDK2
SCHEMBL15739705 0.84 HCRTR1 (0.55) CCR6HCRTR1CCNKCDK2CDK12
SCHEMBL6576773 0.84 NPY5R (0.50) CCR6MAPK1CCNKCDK2CDK12
SCHEMBL3328240 0.83 MAPK1 (0.63) PIM1CCR6HCRTR1MAPK1CCNK
SCHEMBL25258456 0.82 IDH2 (0.56) IDH2CHEK1CCNT1CCNKCCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed