SCHEMBL2015025

SCHEMBL2015025

COc1cc(C(=O)N(C)C(CCNC(=O)c2cccn2C)Cc2ccccc2)ccn1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.70
HCRTR2 O43614 2/20 0.70
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
HRH3 Q9Y5N1 3/20 0.39
KLKB1 P03952 1/20 0.39
PADI4 Q9UM07 3/20 0.38
CTSA P10619 1/20 0.37
KDM5B Q9UGL1 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014960 0.91 HCRTR1 (0.69) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL6919067 0.91 HCRTR1 (0.69) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2017387 0.89 HCRTR1 (0.71) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2016237 0.88 HCRTR1 (0.64) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2054319 0.88 HCRTR1 (0.64) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2052561 0.87 HCRTR1 (0.66) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2014558 0.87 HCRTR1 (0.66) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2016685 0.87 HCRTR1 (0.66) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2012235 0.87 HCRTR1 (0.64) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2014746 0.87 HCRTR1 (0.61) HCRTR1HCRTR2NPC1RAB9AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed