SCHEMBL2015079

SCHEMBL2015079

NC(C=O)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.53
LMNA P02545 1/20 0.53
ALDH1A1 P00352 3/20 0.50
ACP3 P15309 1/20 0.49
ACHE P22303 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
GRM8 O00222 4/20 0.45
GRM4 Q14833 4/20 0.45
NFE2L2 Q16236 1/20 0.45
CA2 P00918 1/20 0.45
CA5A P35218 1/20 0.45
MEN1 O00255 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HSP90AA1 P07900 1/20 0.44
GRM6 O15303 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7062633 0.98 TSHR (0.52) TSHRLMNAALDH1A1ACP3ACHE
SCHEMBL9300488 0.85 TSHR (0.52) TSHRLMNAALDH1A1ACP3ACHE
SCHEMBL2121190 0.82 TSHR (0.61) TSHRLMNAALDH1A1ACP3ACHE
SCHEMBL1701431 0.79 TSHR (0.53) TSHRLMNAALDH1A1ACP3ACHE
SCHEMBL11797282 0.79 TSHR (0.53) TSHRLMNAALDH1A1ACP3ACHE
SCHEMBL2880922 0.79 TSHR (0.53) TSHRLMNAALDH1A1ACP3ACHE
SCHEMBL10522168 0.79 TSHR (0.54) TSHRLMNAALDH1A1TDP1MAPT
SCHEMBL3858019 0.79 TSHR (0.57) TSHRLMNAALDH1A1ACP3ACHE
SCHEMBL6359586 0.79 TSHR (0.57) TSHRLMNAALDH1A1ACP3ACHE
SCHEMBL2433538 0.79 TSHR (0.57) TSHRLMNAALDH1A1ACP3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513098-A1 AMINOPYRIMIDINES AS SYK INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-10-24 EP disclosed
WO-2011075515-A1 AMINOPYRIMIDINES AS SYK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-06-23 WO disclosed