SCHEMBL20153335

SCHEMBL20153335

COC(=O)C(Cc1cnn(CCc2ccc3c(n2)NCCC3)c1)NC(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 19/20 0.55
ITGB6 P18564 17/20 0.55
ITGB3 P05106 2/20 0.45
ITGB1 P05556 1/20 0.41
ITGA5 P08648 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21311528 0.95 ITGAV (0.57) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL20153294 0.88 ITGAV (0.61) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL4194399 0.85 ITGAV (0.61) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL20153293 0.84 ITGAV (0.44) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL4249638 0.84 ITGAV (0.64) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL20153469 0.84 ITGAV (0.64) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL4196182 0.83 ITGAV (0.60) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL20142613 0.82 ITGAV (0.53) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL20153334 0.81 ITGAV (0.67) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL8226900 0.81 ITGAV (0.58) ITGAVITGB6ITGB3ITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed