SCHEMBL20153725

SCHEMBL20153725

CCOC(=O)/C=C/c1cncc(C(C)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.50
DPP4 P27487 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CYP3A4 P08684 2/20 0.48
PTGS2 P35354 1/20 0.47
MAOB P27338 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
FDPS P14324 1/20 0.44
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
RAF1 P04049 2/20 0.41
P2RY12 Q9H244 1/20 0.40
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20153726 0.87 TTR (0.49) TTRDPP4CA12CA1CA2
SCHEMBL21282929 0.85 TTR (0.47) TTRDPP4CA12CA1CA2
SCHEMBL17974436 0.84 CA12 (0.54) TTRDPP4CA12CA1CA2
SCHEMBL7293453 0.81 CA12 (0.51) TTRDPP4CA12CA1CA2
SCHEMBL29278059 0.81 CA12 (0.51) TTRDPP4CA12CA1CA2
SCHEMBL7293458 0.81 CA12 (0.51) TTRDPP4CA12CA1CA2
SCHEMBL29940593 0.81 CA12 (0.51) TTRDPP4CA12CA1CA2
SCHEMBL5991557 0.81 CA12 (0.51) TTRDPP4CA12CA1CA2
SCHEMBL20153870 0.81 HSD17B10 (0.47) TTRDPP4CA12CA1CA2
SCHEMBL18195219 0.80 MAOB (0.56) TTRDPP4CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089357-A1 INDAZOLE DERIVATIVES AS αV INTEGRIN ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed