SCHEMBL20154992

SCHEMBL20154992

CCS(=O)(=O)Cc1ccc(OCC2CC2)c(Br)c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.41
BRD4 O60885 2/20 0.40
PDE4B Q07343 2/20 0.38
HSP90AA1 P07900 1/20 0.38
PDE4A P27815 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
SCN9A Q15858 1/20 0.36
POLB P06746 1/20 0.36
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21191022 0.88 BRD4 (0.50) HRH3BRD4PDE4BPDE4APDE4C
SCHEMBL1439332 0.83 HSP90AA1 (0.47) HRH3PDE4BHSP90AA1POLB
SCHEMBL16658440 0.83 MAPT (0.43)
SCHEMBL3722109 0.78 IKBKE (0.41) HRH3PDE4BPDE4APDE4CPDE4D
SCHEMBL3718807 0.78 HTR2C (0.40) HRH3PDE4BPDE4APDE4CPDE4D
SCHEMBL15067678 0.78 BRD4 (0.49) BRD4POLB
SCHEMBL12891258 0.77 HRH3 (0.39) HRH3PDE4BHSP90AA1PDE4APDE4C
SCHEMBL16651167 0.77 BRD4 (0.50) BRD4HSP90AA1POLBTHRB
SCHEMBL16650725 0.76 BRD4 (0.55) BRD4
SCHEMBL21191023 0.76 HRH3 (0.39) HRH3PDE4BHSP90AA1PDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed