SCHEMBL20156858

SCHEMBL20156858

N#Cc1ccccc1NCCN

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.58
KDM4E B2RXH2 3/20 0.58
HSD17B10 Q99714 2/20 0.58
HPGD P15428 1/20 0.58
CA12 O43570 1/20 0.50
CA3 P07451 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
ALDH1A1 P00352 3/20 0.49
RECQL P46063 1/20 0.49
IDO1 P14902 2/20 0.43
GAA P10253 3/20 0.41
DPP4 P27487 1/20 0.41
FERMT2 Q96AC1 1/20 0.41
NRP1 O14786 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30317451 1.00 TSHR (0.58) TSHRKDM4EHSD17B10HPGDCA12
SCHEMBL17923420 0.81 CA12 (0.50) TSHRKDM4EHSD17B10HPGDCA12
SCHEMBL7528112 0.81 KDM4E (0.58) TSHRKDM4EHSD17B10HPGDALDH1A1
SCHEMBL2122821 0.81 TSHR (0.58) TSHRKDM4EHSD17B10HPGDALDH1A1
SCHEMBL27875640 0.81 KDM4E (0.58) TSHRKDM4EHSD17B10HPGDALDH1A1
SCHEMBL7521970 0.79 KDM4E (0.61) TSHRKDM4EHSD17B10HPGDALDH1A1
SCHEMBL28294998 0.79 CA12 (0.65) TSHRHSD17B10CA12CA3CA4
SCHEMBL3568604 0.78 TSHR (0.56) TSHRKDM4EHSD17B10HPGDALDH1A1
SCHEMBL30528606 0.78 TSHR (0.56) TSHRKDM4EHSD17B10HPGDALDH1A1
SCHEMBL7522731 0.78 KDM4E (0.54) TSHRKDM4EHSD17B10HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115960032-A Aryloxy propanol amine beta-adrenaline receptor ligand with beta-arrestin biased agonistic activity and application thereof 复旦大学 2023-04-14 CN disclosed
EP-3805218-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) Syros Pharmaceuticals, Inc. (US) 2021-04-14 EP disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed