SCHEMBL20157372

SCHEMBL20157372

Cn1cc(-c2cc(CS(C)(=O)=O)ccc2C(=O)c2ccc(F)cc2)c([C@H](CC(=O)OC(C)(C)C)N[SiH]=O)cc1=O

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 10/20 0.39
MAPK14 Q16539 2/20 0.35
BRD2 P25440 2/20 0.31
BRD3 Q15059 2/20 0.31
BRDT Q58F21 2/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362229 0.88 BRD4 (0.39) BRD4MAPK14BRD2BRD3BRDT
SCHEMBL21362230 0.88 BRD4 (0.39) BRD4MAPK14BRD2BRD3BRDT
SCHEMBL21351854 0.79 BRD4 (0.42) BRD4MAPK14BRD2BRD3BRDT
SCHEMBL20158054 0.78 BRD4 (0.41) BRD4MAPK14BRD2BRD3BRDT
SCHEMBL21362189 0.77 BRD4 (0.42) BRD4MAPK14BRD2BRD3BRDT
SCHEMBL21351853 0.76 BRD4 (0.47) BRD4MAPK14BRD2BRD3BRDT
SCHEMBL21351950 0.74 BRD4 (0.35) BRD4MAPK14THRB
SCHEMBL21351914 0.73 BRD4 (0.41) BRD4MAPK14BRD2BRD3BRDT
SCHEMBL21362394 0.73 BRD4 (0.39) BRD4MAPK14THRB
SCHEMBL21352125 0.72 BRD4 (0.34) BRD4MAPK14THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed