SCHEMBL20157431

SCHEMBL20157431

CCSCc1ccc(C(=O)c2ccc(F)cc2)c(-c2cn(C)c(=O)cc2C(C)NS)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.34
MAPT P10636 3/20 0.33
BRD4 O60885 7/20 0.33
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
MAP2K2 P36507 1/20 0.32
MAP2K1 Q02750 1/20 0.32
F11 P03951 1/20 0.31
MAPK14 Q16539 1/20 0.31
POLB P06746 1/20 0.31
ATM Q13315 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ACE P12821 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157715 0.87 BRD4 (0.33) THRBMAPTBRD4ATMHDAC3
SCHEMBL20157434 0.83 BRD4 (0.33) THRBMAPTBRD4MAPK14ATM
SCHEMBL21362394 0.79 BRD4 (0.39) THRBMAPTBRD4ALDH1A1LMNA
SCHEMBL20158149 0.77 GRM5 (0.33) MAPTBRD4LMNAMAP2K2MAP2K1
SCHEMBL21352183 0.76 BRD4 (0.36) THRBMAPTBRD4MAPK14
SCHEMBL21352206 0.76 BRD4 (0.36) THRBMAPTBRD4MAPK14
SCHEMBL21352125 0.75 BRD4 (0.34) THRBMAPTBRD4ALDH1A1LMNA
SCHEMBL21351829 0.74 BRD4 (0.39) THRBMAPTBRD4ATMSMN1; SMN2
SCHEMBL20157691 0.74 MAP2K2 (0.45) THRBMAPTBRD4ALDH1A1LMNA
SCHEMBL21362395 0.74 MAP2K2 (0.43) THRBMAPTALDH1A1LMNAMAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed