SCHEMBL20159989

SCHEMBL20159989

COc1cc(N2C[C@@H]3[C@@H](C)[C@H](C2)[C@H]3N)ncn1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.51
DPP4 P27487 6/20 0.38
DPP8 Q6V1X1 2/20 0.38
DPP7 Q9UHL4 1/20 0.38
LRRK2 Q5S007 4/20 0.36
CYP17A1 P05093 1/20 0.34
DCK P27707 2/20 0.34
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
KCNH2 Q12809 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
APP P05067 1/20 0.33
RIPK1 Q13546 1/20 0.33
ELOVL1 Q9BW60 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18971488 0.81 CYP2C19 (0.47) CYP2C19DPP4DPP8DPP7LRRK2
SCHEMBL21374619 0.81 CYP2C19 (0.52) CYP2C19DPP4DPP8DPP7LRRK2
SCHEMBL18971147 0.81 CYP2C19 (0.52) CYP2C19DPP4DPP8DPP7LRRK2
SCHEMBL18952491 0.81 CYP2C19 (0.52) CYP2C19DPP4DPP8DPP7LRRK2
SCHEMBL18952489 0.81 CYP2C19 (0.52) CYP2C19DPP4DPP8DPP7LRRK2
SCHEMBL21050488 0.81 CYP2C19 (0.52) CYP2C19DPP4DPP8DPP7LRRK2
SCHEMBL23504776 0.81 HRH3 (0.40) DPP4DPP8DPP7CYP17A1PSEN1
SCHEMBL22638877 0.75 CYP2C19 (0.55) CYP2C19DPP4DPP8DPP7LRRK2
SCHEMBL2275882 0.75 CYP2C19 (0.63) CYP2C19CYP17A1DCKRIPK1ELOVL1
Hydrochloric Acid SCHEMBL17077948 0.74 CYP2C19 (0.61) CYP2C19CYP17A1DCKRIPK1ELOVL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed