SCHEMBL20165977

SCHEMBL20165977

O=C1c2ccccc2OC[C@@H]1Br

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.59
MAOB P27338 2/20 0.54
PKM P14618 1/20 0.47
TSHR P16473 1/20 0.47
SIGMAR1 Q99720 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2381366 1.00 CYP19A1 (0.59) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL989344 0.81 CYP19A1 (0.47) CYP19A1MAOBPKMTSHR
SCHEMBL6592452 0.81 CYP19A1 (0.59) CYP19A1MAOBPKMTSHRSIGMAR1
Hydrochloric Acid SCHEMBL697520 0.79 CYP19A1 (0.57) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL18415628 0.78 CYP19A1 (0.61) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL16110707 0.78 CYP19A1 (0.48) CYP19A1
SCHEMBL9094361 0.78 CYP19A1 (0.56) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL7241604 0.77 CYP19A1 (0.59) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL768947 0.77 CYP19A1 (0.59) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL15147097 0.77 CYP19A1 (0.59) CYP19A1MAOBPKMTSHRSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3541812-A1 MGLUR7 AGONIST COMPOUNDS FOR TREATING MGLUR7- REGULATED DISEASES, DISORDERS, OR CONDITIONS Takeda Pharmaceutical Company Limited (JP) 2019-09-25 EP disclosed
WO-2018092921-A1 MGLUR7 AGONIST COMPOUNDS FOR TREATING MGLUR7- REGULATED DISEASES, DISORDERS, OR CONDITIONS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-05-24 WO disclosed