SCHEMBL20169604

SCHEMBL20169604

NCc1ccccc1-c1cncn1F

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.43
IDO1 P14902 10/20 0.37
TDO2 P48775 3/20 0.34
PNMT P11086 2/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
P2RX7 Q99572 1/20 0.33
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170516 0.87 TAAR1 (0.42) IDO1TDO2CYP11B1CYP11B2
SCHEMBL16730945 0.72 CYP11B1 (0.48) IDO1P2RX7CYP11B1CYP11B2
SCHEMBL3787333 0.69 DPP4 (0.73) DPP4PNMTLOXL2
SCHEMBL27519958 0.66 DPP4 (0.61) DPP4PNMT
SCHEMBL27527398 0.65 DPP4 (0.59) DPP4PNMTLOXL2
SCHEMBL25022479 0.64 DPP4 (0.44) DPP4PNMT
SCHEMBL17794539 0.64 DPP4 (0.58) DPP4PNMTLOXL2
SCHEMBL3288611 0.63 DPP4 (0.69) DPP4PNMTLOXL2CYP11B1CYP11B2
SCHEMBL27467061 0.63 DPP4 (0.52) DPP4PNMTCYP11B1CYP11B2
SCHEMBL3288789 0.63 DPP4 (0.62) DPP4TDO2LOXL2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975888-B2 Aryl linked imidazole and triazole derivatives and methods of use thereof for improving the pharmacokinetics of a drug MERCK SHARP & DOHME CORP. (US) 2018-05-22 US disclosed