SCHEMBL20170474

SCHEMBL20170474

CC(c1ccc(F)cc1)n1ccnc1

nearest known ligand 0.90

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 10/20 0.90
CYP19A1 P11511 5/20 0.69
CYP26A1 O43174 3/20 0.62
CYP11B1 P15538 2/20 0.52
CYP11B2 P19099 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16730860 1.00 CYP17A1 (0.90) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL570590 0.83 CYP17A1 (0.67) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL14815347 0.83 CYP11B1 (0.76) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL9664044 0.82 CYP17A1 (0.66) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL16578981 0.82 CYP19A1 (0.69) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL23234111 0.81 CYP17A1 (0.81) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL4043257 0.81 CYP17A1 (0.81) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL10642922 0.81 CYP19A1 (1.00) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL27784193 0.81 CYP17A1 (0.81) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2
SCHEMBL14833233 0.81 CYP17A1 (0.74) CYP17A1CYP19A1CYP26A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed