SCHEMBL20176488

SCHEMBL20176488

Cc1c(F)cc(OC2CN(C)C2)c(F)c1F

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.40
HTR6 P50406 2/20 0.37
HTR2C P28335 4/20 0.34
HTR2B P41595 4/20 0.34
ACACB O00763 4/20 0.33
OXTR P30559 2/20 0.32
SCN1A P35498 1/20 0.30
SCN5A Q14524 1/20 0.30
SCN8A Q9UQD0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20165880 0.86 SLC6A4 (0.41) SLC6A4HTR6HTR2CHTR2BACACB
SCHEMBL20176661 0.83 SLC6A4 (0.44) SLC6A4ACACBOXTRSCN1ASCN8A
SCHEMBL20166170 0.78 SLC6A4 (0.46) SLC6A4HTR6HTR2CHTR2BOXTR
SCHEMBL20165874 0.76 SLC6A4 (0.44) SLC6A4HTR6HTR2CHTR2B
SCHEMBL20176664 0.72 SLC6A4 (0.35) SLC6A4HTR6HTR2CHTR2B
SCHEMBL11288497 0.71 SLC6A2 (0.50) SLC6A4
SCHEMBL20165881 0.71 SLC6A4 (0.60) SLC6A4HTR6HTR2CHTR2BSCN1A
SCHEMBL20068828 0.71 SLC6A4 (0.52) SLC6A4HTR6HTR2CHTR2B
SCHEMBL10261794 0.70 SLC6A2 (0.47) SLC6A4HTR6HTR2CHTR2B
Hydrochloric Acid SCHEMBL20168801 0.70 SLC6A4 (0.34) SLC6A4HTR6HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018091687-A1 NOVEL AZETIDINE DERIVATIVES USEFUL AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION INTEGRATIVE RESEARCH LABORATORIES SWEDEN AB (SE) 2018-05-24 WO disclosed