SCHEMBL20176898

SCHEMBL20176898

COc1cnc(NC(=O)OC(C)(C)C)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
ALOX15 P16050 1/20 0.47
CYP2C19 P33261 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MALT1 Q9UDY8 1/20 0.47
GSK3B P49841 1/20 0.44
DYRK1A Q13627 1/20 0.44
ATR Q13535 1/20 0.43
AAK1 Q2M2I8 5/20 0.42
CHEK1 O14757 2/20 0.41
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
CDK9 P50750 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
MAPKAPK2 P49137 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18308988 0.85 GSK3B (0.47) GSK3BDYRK1AATRAAK1CDK9
SCHEMBL25784199 0.82 ATR (0.57) RAB9ASMN1; SMN2GSK3BDYRK1AATR
SCHEMBL17803539 0.82 ATR (0.48) NPC1TP53RAB9ASMN1; SMN2GSK3B
SCHEMBL28641960 0.82 GSK3B (0.45) NPC1RAB9AGSK3BDYRK1AATR
SCHEMBL25347433 0.81 GSK3B (0.44) NPC1RAB9AGSK3BDYRK1AATR
SCHEMBL2116624 0.81 GSK3B (0.44) GSK3BDYRK1AATRAAK1ALDH1A1
SCHEMBL29954151 0.81 GSK3B (0.44) GSK3BDYRK1AATRAAK1CHEK1
SCHEMBL15354547 0.81 GSK3B (0.44) GSK3BDYRK1AATRAAK1ALDH1A1
SCHEMBL22448769 0.80 GSK3B (0.43) CYP3A4GSK3BDYRK1AATRAAK1
SCHEMBL30381133 0.80 ATR (0.54) SMN1; SMN2GSK3BDYRK1AATRAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed
WO-2018092047-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE JOINT STOCK COMPANY "BIOCAD" (RU) 2018-05-24 WO disclosed