SCHEMBL20176931

SCHEMBL20176931

Cc1c(C(CNC(=O)OC(C)(C)C)NS(=O)(=O)CCCCl)ccc2c1COC2=O

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 20/20 0.39
KCNH2 Q12809 5/20 0.39
ACHE P22303 1/20 0.39
SSTR1 P30872 1/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21265975 1.00 KCNJ1 (0.39) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL20168135 0.89 KCNJ1 (0.43) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL20168133 0.89 KCNJ1 (0.43) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL21266199 0.88 KCNJ1 (0.45) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL20176984 0.88 KCNJ1 (0.45) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL21265973 0.86 KCNJ1 (0.40) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL21265947 0.83 KCNJ1 (0.48) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL20177025 0.83 KCNJ1 (0.48) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL21265960 0.83 KCNJ1 (0.49) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL21265972 0.83 KCNJ1 (0.46) KCNJ1KCNH2ACHESSTR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139862-B Substituted bicyclic heterocyclic derivatives useful as ROMK channel inhibitors 百时美施贵宝公司 2024-01-16 CN disclosed
WO-2018093569-A1 SUBSTITUTED BICYCLE HETEROCYCLIC DERIVATIVES USEFUL AS ROMK CHANNEL INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-24 WO disclosed