SCHEMBL20179753

SCHEMBL20179753

COC(=O)c1ccc(OC2CCN(CCCF)C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 15/20 0.53
AGTR2 P50052 1/20 0.49
ESR2 Q92731 1/20 0.48
CCR1 P32246 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20179622 1.00 ESR1 (0.53) ESR1AGTR2ESR2CCR1
SCHEMBL29756809 0.88 HRH2 (0.56) ESR1AGTR2ESR2
SCHEMBL20165868 0.87 ESR1 (0.61) ESR1AGTR2ESR2
SCHEMBL20165122 0.87 ESR1 (0.61) ESR1AGTR2ESR2
SCHEMBL20165121 0.86 ESR1 (0.54) ESR1AGTR2ESR2
SCHEMBL20165124 0.86 ESR1 (0.54) ESR1AGTR2ESR2
Hydrochloric Acid SCHEMBL29756830 0.86 ESR1 (0.60) ESR1AGTR2ESR2
Hydrochloric Acid SCHEMBL29756701 0.85 ESR1 (0.53) ESR1AGTR2ESR2
SCHEMBL20165047 0.84 ESR1 (0.49) ESR1AGTR2ESR2
SCHEMBL20165045 0.84 ESR1 (0.49) ESR1AGTR2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018091153-A1 NOVEL SUBSTITUTED N-(3-FLUOROPROPYL)-PYRROLIDINE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF SANOFI (FR) 2018-05-24 WO disclosed