SCHEMBL20180817

SCHEMBL20180817

COc1ccc(N2CCOC2=O)cc1I

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.46
MTOR P42345 1/20 0.46
PDE10A Q9Y233 1/20 0.41
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39
LRRK2 Q5S007 2/20 0.39
MIF P14174 1/20 0.38
APLNR P35414 1/20 0.37
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
SLC9A3 P48764 1/20 0.35
MMP12 P39900 2/20 0.35
MMP13 P45452 2/20 0.35
LMNA P02545 1/20 0.35
SCN9A Q15858 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA7 P43166 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17151142 0.84 PIK3CA (0.47) PIK3CAMTORPDE10ACCNCCDK8
SCHEMBL12445267 0.83 PIK3CA (0.46) PIK3CAMTORPDE10ALRRK2MIF
SCHEMBL30884507 0.81 PIK3CA (0.47) PIK3CAMTORPDE10ACCNCCDK8
SCHEMBL15651208 0.81 PIK3CA (0.47) PIK3CAMTORPDE10ACCNCCDK8
SCHEMBL20180814 0.81 F10 (0.47) MTORLRRK2
SCHEMBL21376420 0.81 PIK3CA (0.44) PIK3CAMTORPDE10ACCNCCDK8
SCHEMBL17148220 0.81 PIK3CA (0.44) PIK3CAMTORPDE10ACCNCCDK8
SCHEMBL30602385 0.80 PIK3CA (0.46) PIK3CAMTORPDE10ACCNCCDK8
SCHEMBL9997046 0.80 PIK3CA (0.46) PIK3CAMTORPDE10ACCNCCDK8
SCHEMBL14146011 0.80 PIK3CA (0.46) PIK3CAMTORPDE10ACCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093579-A1 TRIAZOLE PHENYL COMPOUNDS AS AGONISTS OF THE APJ RECEPTOR AMGEN INC. (US) 2018-05-24 WO disclosed