SCHEMBL20181901

SCHEMBL20181901

CC(c1cnc(-c2ccccc2F)[nH]1)n1cc(C(=N)/C=C\N)c2c(N)ncnc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 9/20 0.35
KDR P35968 8/20 0.35
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
PRKDC P78527 2/20 0.33
SRC P12931 6/20 0.33
LCK P06239 4/20 0.33
TEK Q02763 3/20 0.33
MTOR P42345 2/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
HCK P08631 1/20 0.33
EPHB4 P54760 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
PDPK1 O15530 3/20 0.32
AKT1 P31749 1/20 0.32
NTRK1 P04629 1/20 0.32
NTRK3 Q16288 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182216 0.83 KDR (0.40) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL20162795 0.82 KDR (0.42) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL20173304 0.82 KDR (0.40) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL30036859 0.82 KDR (0.42) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL20175297 0.78 KDR (0.42) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL20175447 0.78 KDR (0.40) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL20175829 0.78 KDR (0.43) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL30892139 0.78 KDR (0.40) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL20173308 0.77 KDR (0.42) RETKDRPIK3CDPIK3CAPIK3CB
SCHEMBL20162933 0.77 PIK3CD (0.43) RETKDRPIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed