SCHEMBL20182176

SCHEMBL20182176

Cc1cn(C(C)c2cc(-c3ccccc3F)no2)c2ncnc(N)c12

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RET P07949 16/20 0.46
CFTR P13569 1/20 0.40
KDR P35968 3/20 0.38
SRC P12931 2/20 0.38
EGFR P00533 1/20 0.38
CDK1 P06493 1/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
PRKDC P78527 1/20 0.38
LCK P06239 1/20 0.37
TEK Q02763 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162767 0.89 RET (0.45) RETCFTRKDRSRCPIK3CD
SCHEMBL30037388 0.89 RET (0.45) RETCFTRKDRSRCPIK3CD
SCHEMBL20173323 0.89 RET (0.45) RETCFTRKDRSRCPIK3CD
SCHEMBL30538106 0.85 KDR (0.46) RETKDRSRCEGFRPIK3CD
SCHEMBL30037546 0.85 KDR (0.46) RETKDRSRCEGFRPIK3CD
SCHEMBL20162651 0.85 KDR (0.46) RETKDRSRCEGFRPIK3CD
SCHEMBL20162649 0.85 KDR (0.46) RETKDRSRCEGFRPIK3CD
SCHEMBL20162640 0.84 RET (0.46) RETCFTRKDRSRCEGFR
SCHEMBL20162645 0.84 RET (0.46) RETCFTRKDRSRCEGFR
SCHEMBL20173328 0.84 KDR (0.45) RETKDRSRCEGFRPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed