SCHEMBL20182285

SCHEMBL20182285

CCC(/C(=C/Nc1cccc(F)c1F)N=N)n1cc(-c2cnc(C(F)(F)F)nc2)c2c(N)ncnc21

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CFTR P13569 7/20 0.41
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
PRKDC P78527 1/20 0.37
SRC P12931 5/20 0.35
ABL1 P00519 2/20 0.35
EGFR P00533 2/20 0.35
ABL2 P42684 2/20 0.35
EIF2AK3 Q9NZJ5 3/20 0.34
KDR P35968 1/20 0.33
TEK Q02763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182197 0.94 CFTR (0.43) CFTRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL20182294 0.90 CFTR (0.40) CFTRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL20181910 0.90 CFTR (0.38) CFTRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL20182296 0.88 CFTR (0.41) CFTRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL20182225 0.87 CFTR (0.39) CFTRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL20182355 0.85 CFTR (0.38) CFTR
SCHEMBL20182269 0.85 CFTR (0.38) CFTR
SCHEMBL20182255 0.84 SRC (0.39) CFTRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL20182362 0.84 CFTR (0.40) CFTRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL20181912 0.82 SRC (0.41) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed