SCHEMBL20182825

SCHEMBL20182825

CC(C(=O)NC1COc2ccccc2C1O)c1ccccc1

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 9/20 0.75
LTB4R Q15722 4/20 0.44
LTB4R2 Q9NPC1 4/20 0.44
P2RX7 Q99572 2/20 0.42
TRPM8 Q7Z2W7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21542318 1.00 GRM7 (0.75) GRM7LTB4RLTB4R2P2RX7TRPM8
SCHEMBL20165981 1.00 GRM7 (0.75) GRM7LTB4RLTB4R2P2RX7TRPM8
SCHEMBL21542320 1.00 GRM7 (0.75) GRM7LTB4RLTB4R2P2RX7TRPM8
SCHEMBL20165982 1.00 GRM7 (0.75) GRM7LTB4RLTB4R2P2RX7TRPM8
SCHEMBL20165979 1.00 GRM7 (0.75) GRM7LTB4RLTB4R2P2RX7TRPM8
SCHEMBL21542214 0.90 GRM7 (0.76) GRM7LTB4RLTB4R2P2RX7
SCHEMBL21542216 0.90 GRM7 (0.76) GRM7LTB4RLTB4R2P2RX7
SCHEMBL20182770 0.90 GRM7 (0.76) GRM7LTB4RLTB4R2P2RX7
SCHEMBL21542206 0.86 GRM7 (0.61) GRM7LTB4RLTB4R2P2RX7TRPM8
SCHEMBL21542241 0.86 GRM7 (0.61) GRM7LTB4RLTB4R2P2RX7TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3541812-B1 MGLUR7 AGONIST COMPOUNDS FOR TREATING MGLUR7- REGULATED DISEASES, DISORDERS, OR CONDITIONS TAKEDA PHARMACEUTICALS CO (JP) 2023-06-14 EP disclosed
WO-2018092921-A1 MGLUR7 AGONIST COMPOUNDS FOR TREATING MGLUR7- REGULATED DISEASES, DISORDERS, OR CONDITIONS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-05-24 WO disclosed