SCHEMBL20183010

SCHEMBL20183010

Cn1ncc(Cn2cccn2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
PDE4B Q07343 2/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HTT P42858 1/20 0.36
TSHR P16473 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ADCY10 Q96PN6 1/20 0.35
BRD4 O60885 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
TDP1 Q9NUW8 1/20 0.33
DAO P14920 1/20 0.33
FDPS P14324 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1908658 0.72
SCHEMBL24017979 0.70 CYP11B1 (0.49) MAPT
SCHEMBL17489171 0.69 PDE4B (0.48) GAAMAPTNOS3NOS1PDE4B
SCHEMBL28858185 0.69 GAA (0.46) GAAMAPTNOS3NOS1PDE4B
SCHEMBL16260559 0.69 GAA (0.46) GAAMAPTNOS3NOS1PDE4B
SCHEMBL12945953 0.69
SCHEMBL28416242 0.69
SCHEMBL6002309 0.68 GAA (0.49) GAAMAPTNOS3NOS1HDAC1
SCHEMBL28205957 0.67 CYP11B1 (0.49) GAAMAPTNOS3NOS1HDAC1
SCHEMBL19260079 0.67 MAPT (0.47) GAAMAPTHDAC1HDAC6HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092921-A1 MGLUR7 AGONIST COMPOUNDS FOR TREATING MGLUR7- REGULATED DISEASES, DISORDERS, OR CONDITIONS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-05-24 WO disclosed