SCHEMBL20184255

SCHEMBL20184255

Cc1c(C(O)CN2CCC3(CC2)CCN(c2ccc(C#N)cn2)CC3)ccc2c1COC2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 20/20 1.00
KCNH2 Q12809 4/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16438723 1.00 KCNJ1 (1.00) KCNJ1KCNH2
SCHEMBL17925120 0.95 KCNJ1 (1.00) KCNJ1KCNH2
SCHEMBL16438733 0.95 KCNJ1 (1.00) KCNJ1KCNH2
SCHEMBL17925088 0.95 KCNJ1 (1.00) KCNJ1KCNH2
SCHEMBL16438931 0.95 KCNJ1 (1.00) KCNJ1KCNH2
SCHEMBL17925108 0.94 KCNJ1 (1.00) KCNJ1KCNH2
SCHEMBL16438746 0.94 KCNJ1 (1.00) KCNJ1KCNH2
SCHEMBL14919331 0.93 KCNJ1 (0.86) KCNJ1KCNH2
SCHEMBL14919329 0.93 KCNJ1 (0.86) KCNJ1KCNH2
SCHEMBL16438944 0.90 KCNJ1 (1.00) KCNJ1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3027625-B1 SPIRO-FUSED DERIVATIVES OF PIPERIDINE USEFUL FOR THE TREATMENT OF INTER ALIA HYPERTENSION AND ACUTE OR CHRONIC HEART FAILURE MERCK SHARP & DOHME (US) 2018-05-30 EP disclosed