SCHEMBL20187758

SCHEMBL20187758

CSc1cnc(Nc2ccc(C(=O)Nc3cccc(CN(C)C)c3)cc2)nc1-c1ccc(C#N)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.48
PDGFRB P09619 1/20 0.48
BCR P11274 1/20 0.48
PDGFRA P16234 1/20 0.48
PRKCA P17252 1/20 0.48
ROCK2 O75116 2/20 0.46
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
CDK7 P50613 2/20 0.41
CCNH P51946 2/20 0.41
CYP19A1 P11511 1/20 0.41
CAMK2D Q13557 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
AURKA O14965 1/20 0.40
CDK2 P24941 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21799061 0.88 ABL1 (0.41) ABL1PDGFRBBCRPDGFRAPRKCA
SCHEMBL30114760 0.88 ABL1 (0.41) ABL1PDGFRBBCRPDGFRAPRKCA
SCHEMBL22503491 0.86 ABL1 (0.49) ABL1PDGFRBBCRPDGFRAPRKCA
SCHEMBL21799077 0.81
SCHEMBL20187902 0.79 TRPV1 (0.52) ABL1PDGFRBBCRPDGFRAPRKCA
SCHEMBL30530305 0.79 TRPV1 (0.52) ABL1PDGFRBBCRPDGFRAPRKCA
SCHEMBL20188166 0.78 AURKA (0.44) ABL1PDGFRBPDGFRAAURKA
SCHEMBL30530307 0.78 AURKA (0.44) ABL1PDGFRBPDGFRAAURKA
SCHEMBL21799125 0.77 PIKFYVE (0.43) TRPV1
SCHEMBL21799092 0.76 TRPV1 (0.51) ABL1PDGFRBBCRPDGFRAPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544685-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF Development Center for Biotechnology (TW) 2019-10-02 EP disclosed
WO-2018098250-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 2018-05-31 WO disclosed