SCHEMBL20190171

SCHEMBL20190171

CCc1ccc(COC(=O)N2CC[C@@H](CNc3ncccn3)C(F)(F)C2)cc1

nearest known ligand 0.86

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 17/20 0.86
KCNH2 Q12809 3/20 0.63
CYP2D6 P10635 2/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20202786 1.00 GRIN2B (0.86) GRIN2BKCNH2CYP2D6
SCHEMBL21404307 1.00 GRIN2B (0.86) GRIN2BKCNH2CYP2D6
SCHEMBL20190803 0.97 GRIN2B (0.82) GRIN2BKCNH2CYP2D6
SCHEMBL20190802 0.97 GRIN2B (0.82) GRIN2BKCNH2CYP2D6
SCHEMBL18280950 0.93 GRIN2B (1.00) GRIN2BKCNH2CYP2D6
SCHEMBL20190220 0.93 GRIN2B (1.00) GRIN2BKCNH2CYP2D6
SCHEMBL18280951 0.93 GRIN2B (1.00) GRIN2BKCNH2CYP2D6
SCHEMBL20189499 0.91 GRIN2B (0.84) GRIN2BKCNH2CYP2D6
SCHEMBL21404297 0.91 GRIN2B (0.84) GRIN2BKCNH2CYP2D6
SCHEMBL20202990 0.91 GRIN2B (0.84) GRIN2BKCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544610-A1 TREATMENT OF AUTISM SPECTRUM DISORDERS, OBSESSIVE-COMPULSIVE DISORDER AND ANXIETY DISORDERS Rugen Holdings (Cayman) Limited (KY) 2019-10-02 EP disclosed
WO-2018098128-A1 TREATMENT OF AUTISM SPECTRUM DISORDERS, OBSESSIVE-COMPULSIVE DISORDER AND ANXIETY DISORDERS RUGEN HOLDINGS (CAYMAN) LIMITED (KY) 2018-05-31 WO disclosed