SCHEMBL20197290

SCHEMBL20197290

CCCc1ccc(I)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30
IDO1 P14902 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA5 P31644 1/20 0.30
GABRA3 P34903 1/20 0.30
GABRA2 P47869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9706383 0.86 KCNH2 (0.46) KDM4ELMNACYP3A4GABRPGABRD
SCHEMBL9850704 0.84 KCNH2 (0.48) KDM4ELMNACYP3A4GABRPGABRD
SCHEMBL9697516 0.84 KCNH2 (0.48) KDM4ELMNACYP3A4GABRPGABRD
SCHEMBL9706417 0.84 KCNH2 (0.48) KDM4ELMNACYP3A4GABRPGABRD
SCHEMBL9850711 0.84 KCNH2 (0.48) KDM4ELMNACYP3A4GABRPGABRD
SCHEMBL1022641 0.82
SCHEMBL19313500 0.79 MYC (0.35) HRH3CYP1A2CYP2D6
SCHEMBL19313495 0.78 PDE2A (0.34)
SCHEMBL991122 0.76 CCR1 (0.46) HRH3KDM4ELMNACYP3A4TSHR
SCHEMBL16389875 0.76 HRH3 (0.47) HRH3KDM4ELMNACYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed