SCHEMBL20204049

SCHEMBL20204049

CCCCC(CCO)C(=O)NNc1cnc(-c2ccc(OC(F)(F)F)cc2)cn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.56
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
ADORA3 P0DMS8 1/20 0.37
ABL1 P00519 3/20 0.36
PPARD Q03181 2/20 0.35
GRIN2B Q13224 1/20 0.35
ALOX5 P09917 1/20 0.35
PPARG P37231 1/20 0.35
TSHR P16473 1/20 0.35
SCN10A Q9Y5Y9 2/20 0.35
SCN2A Q99250 1/20 0.35
CXCR2 P25025 1/20 0.35
AHR P35869 1/20 0.35
BCR P11274 2/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
VNN1 O95497 1/20 0.34
DGAT1 O75907 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20203824 0.81 CYP1A2 (0.67) CYP1A2ADORA3ABL1PPARDGRIN2B
SCHEMBL20203902 0.78 CYP1A2 (0.71) CYP1A2ADORA3ABL1PPARDGRIN2B
SCHEMBL20203801 0.75 CYP1A2 (0.67) CYP1A2HDAC3HDAC1HDAC2ADORA3
SCHEMBL20189734 0.75 CYP1A2 (0.61) CYP1A2HDAC3HDAC1HDAC2ADORA3
SCHEMBL20204022 0.73 CYP1A2 (0.69) CYP1A2ADORA3ABL1GRIN2BSCN10A
SCHEMBL20191119 0.72 CYP1A2 (1.00) CYP1A2ADORA3ABL1GRIN2BSCN10A
SCHEMBL23571890 0.69 CYP1A2 (0.69) CYP1A2ADORA3ABL1GRIN2BSCN10A
SCHEMBL26031183 0.69 CYP1A2 (0.44) CYP1A2DGAT1
SCHEMBL23571203 0.69 CYP1A2 (0.57) CYP1A2ADORA3ABL1SCN10ASCN2A
SCHEMBL20190030 0.68 CYP1A2 (0.63) CYP1A2HDAC1HDAC2ADORA3ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018098499-A1 COMPOUNDS AND THEIR METHODS OF USE PRAXIS PRECISION MEDICINES, INC. (US) 2018-05-31 WO disclosed