SCHEMBL20207260

SCHEMBL20207260

Cc1oc(=O)oc1COC(=O)[C@H](CCC(=O)O)NC(=O)c1ccc(CCc2c[nH]c3nc(N)[nH]c(=O)c23)cc1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TYMS P04818 9/20 0.70
DHFR P00374 6/20 0.70
FOLR1 P15328 6/20 0.70
SLC46A1 Q96NT5 6/20 0.70
SLC19A1 P41440 5/20 0.70
GART P22102 5/20 0.70
ATIC P31939 2/20 0.70
FOLR2 P14207 2/20 0.70
SHMT1 P34896 1/20 0.70
FRK P42685 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20207261 1.00 TYMS (0.70) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL20207269 0.94 TYMS (0.61) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL20207506 0.94 TYMS (0.60) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL20207405 0.92 TYMS (0.59) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL20207399 0.92 TYMS (0.59) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL20207398 0.89 TYMS (0.55) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL1302274 0.87 TYMS (0.79) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL1302278 0.87 TYMS (0.79) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL15078861 0.86 GART (0.84) TYMSDHFRFOLR1SLC46A1SLC19A1
SCHEMBL22326828 0.85 GART (0.77) TYMSDHFRFOLR1SLC46A1SLC19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096853-A1 NOVEL MEDOXOMIL AND HEMIACETAL ESTERS OF PEMETREXED, PRODUCTION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION CONTAINING ESTER PRODRUG 学校法人近畿大学 2018-05-31 WO disclosed