Predicted protein targets (top 16)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | SCN5A | Q14524 | 14/20 | 0.45 |
| ▸ | SCN1A | P35498 | 2/20 | 0.41 |
| ▸ | SCN2A | Q99250 | 2/20 | 0.41 |
| ▸ | CACNA2D1 | P54289 | 1/20 | 0.39 |
| ▸ | KDM4E | B2RXH2 | 1/20 | 0.39 |
| ▸ | NPC1 | O15118 | 1/20 | 0.39 |
| ▸ | ALDH1A1 | P00352 | 1/20 | 0.39 |
| ▸ | GAA | P10253 | 1/20 | 0.39 |
| ▸ | MAPT | P10636 | 1/20 | 0.39 |
| ▸ | RAB9A | P51151 | 1/20 | 0.39 |
| ▸ | KCNH2 | Q12809 | 1/20 | 0.37 |
| ▸ | SCN10A | Q9Y5Y9 | 1/20 | 0.37 |
| ▸ | RXRA | P19793 | 1/20 | 0.36 |
| ▸ | GRIN1 | Q05586 | 1/20 | 0.36 |
| ▸ | GRIN2B | Q13224 | 1/20 | 0.36 |
| ▸ | MCHR1 | Q99705 | 1/20 | 0.36 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL20209001 | 0.78 | SCN5A (0.52) | SCN5ASCN1ASCN2AKDM4ENPC1 | |
| SCHEMBL20190662 | 0.78 | SCN5A (0.47) | SCN5ASCN1ASCN2AKDM4ENPC1 | |
| SCHEMBL20190225 | 0.78 | SCN5A (0.50) | SCN5ASCN1ASCN2AKDM4ENPC1 | |
| SCHEMBL20189412 | 0.74 | GRM5 (0.48) | SCN5AKDM4ENPC1ALDH1A1GAA | |
| SCHEMBL23572498 | 0.73 | SCN5A (0.52) | SCN5ASCN1ASCN2AKDM4ENPC1 | |
| SCHEMBL20208519 | 0.73 | SCN5A (0.71) | SCN5ASCN1ASCN2AKDM4ENPC1 | |
| SCHEMBL26539098 | 0.72 | SCN5A (0.52) | SCN5ASCN1ASCN2AKDM4ENPC1 | |
| SCHEMBL20203710 | 0.71 | SCN5A (0.65) | SCN5ASCN1ASCN2A | |
| SCHEMBL20209224 | 0.71 | SCN5A (0.56) | SCN5ASCN1ASCN2A | |
| SCHEMBL9061989 | 0.69 | CHRM5 (0.46) | SCN5ASCN1ASCN2AKCNH2SCN10A |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| WO-2018098500-A1 | COMPOUNDS AND THEIR METHODS OF USE | PRAXIS PRECISION MEDICINES, INC. (US) | 2018-05-31 | — | — | WO | disclosed |